SCHEMBL7759833

SCHEMBL7759833

CN1C[S+]([O-])c2cc(CCCN3CCOCC3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.51
POLB P06746 1/20 0.50
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
HTR2A P28223 1/20 0.38
SCN1A P35498 1/20 0.38
HTR2B P41595 1/20 0.38
KCNH2 Q12809 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
LSS P48449 1/20 0.38
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449991 0.96 SIGMAR1 (0.47) SIGMAR1POLBHTTKMT2ATHRA
SCHEMBL8948173 0.90 SIGMAR1 (0.46) SIGMAR1HRH3
SCHEMBL8948263 0.88 SIGMAR1 (0.48) SIGMAR1CHRM2KCNH2HRH3
SCHEMBL8948349 0.86 SLC6A4 (0.37) SIGMAR1POLBHRH3
SCHEMBL9449597 0.81 SIGMAR1 (0.55) SIGMAR1CYP1A2LMNA
SCHEMBL9230596 0.80 SIGMAR1 (0.54) SIGMAR1POLBCYP1A2
SCHEMBL7759855 0.80 CCR3 (0.58) SIGMAR1KMT2AALDH1A1HTR2B
SCHEMBL9684037 0.80 S1PR1 (0.38) SIGMAR1THRATHRBALDH1A1CHRM2
SCHEMBL7760492 0.80
SCHEMBL9684946 0.79 BCHE (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673934-B1 Aminoalkyl benzothiazolinones, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-04-25 EP claimed
US-5512569-A SIGMA RECEPTOR DISORDERS; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 1996-04-30 US claimed
EP-0673934-A1 Aminoalkyl benzothiazolinones, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1995-09-27 EP claimed
US-5512569-A SIGMA RECEPTOR DISORDERS; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 1996-04-30 US disclosed