SCHEMBL7765719

SCHEMBL7765719

CCCCC(=O)[N]NC(=O)C(Cl)(Cl)Cl

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
TP53 P04637 1/20 0.39
CES1 P23141 6/20 0.37
CES2 O00748 5/20 0.37
CA1 P00915 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.32
EPHX1 P07099 1/20 0.31
FAAH O00519 2/20 0.31
HSP90AA1 P07900 1/20 0.31
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7771366 0.89 TSHR (0.34) CES1CES2TSHR
SCHEMBL7769364 0.81 EPHX1 (0.46) ALDH1A1CES1CES2EPHX1FAAH
SCHEMBL7770033 0.80 L3MBTL1 (0.32)
SCHEMBL7769447 0.76 FAAH (0.42) ALDH1A1TP53CES1CES2CA1
SCHEMBL7771405 0.74 ALDH1A1 (0.39) ALDH1A1TP53CES1CES2CA1
SCHEMBL7770041 0.73 CES1 (0.39) ALDH1A1TP53CES1CES2CA1
SCHEMBL7769845 0.73 FAAH (0.46) ALDH1A1TP53CES1CES2MAPT
SCHEMBL7771427 0.72 CES1 (0.38) ALDH1A1TP53CES1CES2CA1
SCHEMBL7766040 0.72 CES1 (0.38) ALDH1A1TP53CES1CES2CA1
SCHEMBL7765980 0.70 CES2 (0.41) ALDH1A1TP53CES1CES2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765879-B1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO CO (JP) 2001-02-14 EP disclosed
US-5861429-A MITICIDES AND ANTHELMINTICS SANKYO COMPANY, LIMITED (JP) 1999-01-19 US disclosed
EP-0765879-A1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO COMPANY LIMITED (JP) 1997-04-02 EP disclosed