SCHEMBL7766463

SCHEMBL7766463

COc1ccccc1N1CCN(Cc2ccc3c(c2)[S+]([O-])CN3C)CC1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.61
MAPK1 P28482 1/20 0.60
DRD4 P21917 5/20 0.58
ALDH1A1 P00352 2/20 0.57
KDM4E B2RXH2 3/20 0.56
KMT2A Q03164 1/20 0.56
DRD2 P14416 6/20 0.56
DRD3 P35462 4/20 0.56
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
TSHR P16473 1/20 0.54
HRH2 P25021 1/20 0.53
HRH1 P35367 1/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9449688 0.90 ADRA1D (0.61) DRD2
SCHEMBL7761667 0.89 DRD2 (0.60) DRD2DRD3
SCHEMBL7762716 0.84 KDM4E (0.56) MAPK1DRD4ALDH1A1KDM4EDRD2
Hydrochloric Acid SCHEMBL8406359 0.83 KDM4E (0.55) MAPK1DRD4ALDH1A1KDM4EDRD2
SCHEMBL7767380 0.82 DRD4 (0.53) DRD4ALDH1A1KDM4EKMT2ADRD2
SCHEMBL8621656 0.81 KDM4E (0.61) DRD4ALDH1A1KDM4EDRD2DRD3
SCHEMBL7762764 0.77 KDM4E (0.55) DRD4ALDH1A1KDM4EDRD2DRD3
SCHEMBL9225440 0.76 MAPK1 (0.81) HTR7MAPK1DRD4ALDH1A1KDM4E
SCHEMBL9720648 0.76 HTR7 (0.70) HTR7MAPK1DRD4ALDH1A1KDM4E
SCHEMBL6031061 0.76 MAPK1 (0.80) HTR7MAPK1DRD4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP claimed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US claimed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP claimed
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP disclosed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US disclosed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed