SCHEMBL8621656

SCHEMBL8621656

COc1cccc(N2CCN(Cc3ccc4c(c3)[S+]([O-])CN4C)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.61
ALDH1A1 P00352 3/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
MAPT P10636 2/20 0.58
TSHR P16473 2/20 0.58
GFER P55789 1/20 0.54
KCNH2 Q12809 2/20 0.53
DRD2 P14416 2/20 0.53
SIGMAR1 Q99720 1/20 0.49
TP53 P04637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
GAA P10253 1/20 0.48
CASP1 P29466 1/20 0.47
CASP4 P49662 1/20 0.47
CASP5 P51878 1/20 0.47
DRD4 P21917 2/20 0.45
DRD3 P35462 1/20 0.45
HTR1A P08908 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7767380 0.90 DRD4 (0.53) KDM4EALDH1A1SMN1; SMN2MAPTTSHR
SCHEMBL7766463 0.81 HTR7 (0.61) KDM4EALDH1A1TSHRDRD2DRD4
SCHEMBL7762764 0.81 KDM4E (0.55) KDM4EALDH1A1SMN1; SMN2MAPTDRD2
SCHEMBL8570664 0.77 SIGMAR1 (0.81) KDM4EALDH1A1SMN1; SMN2MAPTTSHR
SCHEMBL7765506 0.77 CA2 (0.46) KDM4EALDH1A1SMN1; SMN2
SCHEMBL7762716 0.76 KDM4E (0.56) KDM4EALDH1A1SMN1; SMN2TSHRDRD2
SCHEMBL25370948 0.76 KDM4E (0.80) KDM4EALDH1A1SMN1; SMN2MAPTTSHR
SCHEMBL6031705 0.76 KDM4E (1.00) KDM4EALDH1A1SMN1; SMN2MAPTTSHR
SCHEMBL27395515 0.76 KDM4E (0.80) KDM4EALDH1A1SMN1; SMN2MAPTTSHR
Hydrochloric Acid SCHEMBL8406359 0.76 KDM4E (0.55) KDM4EALDH1A1SMN1; SMN2TSHRDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed