SCHEMBL7767017

SCHEMBL7767017

C=CSc1ccc(C)cc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 1/20 0.40
TP53 P04637 3/20 0.38
TDP1 Q9NUW8 3/20 0.38
HTR1A P08908 7/20 0.36
HTR3A P46098 7/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
LMNA P02545 2/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23795423 0.83 LMNA (0.39) TP53TDP1LMNAHPGDMEN1
SCHEMBL20647862 0.81 TP53 (0.47) HAO1TP53TDP1HTR1AHTR3A
SCHEMBL21553822 0.79 ALDH1A1 (0.31) HPGDMAPTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL29543901 0.79 ALDH1A1 (0.31) HPGDMAPTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL26062395 0.76 TRPA1 (0.35) LMNAGAAMAPTALOX12HSD17B10
SCHEMBL13840027 0.75 NPC1 (0.53) TP53TDP1LMNAHPGDMEN1
SCHEMBL1145702 0.75 HAO1 (0.43) HAO1TP53TDP1HTR1AHTR3A
SCHEMBL29475022 0.74 HAO1 (0.55) HAO1TP53TDP1HTR1AHTR3A
SCHEMBL76793 0.74 HAO1 (0.55) HAO1TP53TDP1HTR1AHTR3A
SCHEMBL29411684 0.74 NPC1 (0.50) HAO1TP53TDP1HTR1AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019157050-A1 CERTAIN (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES FOR TREATING ANCA ASSOCIATED VASCULITIDES INSMED INCORPORATED (US) 2019-08-15 WO disclosed
EP-2791137-B1 PYRAZOLOPYRIDINE DERIVATIVES, PREPARATION PROCESS THEREFOR AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2019-01-23 EP disclosed
EP-0711813-B1 Antifouling coating composition HITACHI CHEMICAL CO LTD (JP) 2001-07-25 EP disclosed
US-5773508-A BIODEGRADABLE POLYMER OF ADDITION COPOLYMERS FOR PROTECTIVE COATINGS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-06-30 US disclosed
EP-0711813-A2 Coating varnish composition and antifouling coating composition Hitachi Chemical Co., Ltd. (JP) 1996-05-15 EP disclosed