Sulfotep

Sulfotep

SCHEMBL7767701

CCCC(=O)O.CCOP(=S)(OCC)OP(=S)(OCC)OCC

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR3 O14843 1/20 0.52
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
AKR1B1 P15121 1/20 0.37
GPR84 Q9NQS5 7/20 0.35
PPARG P37231 7/20 0.35
PPARD Q03181 7/20 0.35
PPARA Q07869 7/20 0.35
HDAC11 Q96DB2 5/20 0.35
TSHR P16473 4/20 0.35
PTPN1 P18031 3/20 0.35
ALDH1A1 P00352 3/20 0.35
TLR2 O60603 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
FABP4 P15090 2/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfotep SCHEMBL1163295 1.00 FFAR3 (0.52) FFAR3HDAC3HDAC1HDAC2HDAC8
Sulfotep SCHEMBL1163969 0.89 AKR1B1 (0.48) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL2026147 0.88 AKR1B1 (0.46) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL1163364 0.87 AKR1B1 (0.57) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL2336663 0.86 GPR84 (0.48) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL2786434 0.86 GPR84 (0.48) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL8472533 0.85 GPR84 (0.59) AKR1B1GPR84PPARGPPARDPPARA
Sulfotep SCHEMBL1163901 0.85 FFAR3 (0.46) FFAR3PPARDTSHRALDH1A1TDP1
Sulfotep SCHEMBL7762968 0.85 FFAR3 (0.46) FFAR3PPARDTSHRALDH1A1TDP1
Sulfotep SCHEMBL461502 0.85 TDP1 (0.39) PPARDTSHRALDH1A1TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310161-B1 ACRYLATE WITH MONOTHIOL AND CONJUGATED AROMATIC COMPOUND UCB S.A. (BE) 2001-10-30 US disclosed
EP-0810992-B1 SULFUR-CONTAINING COMPOUNDS FOR OPTICAL GRADE POLYMERIC CASTING COMPOSITIONS UCB SA (BE) 2001-06-13 EP disclosed
US-6051733-A Sulfur-containing compounds for optical grade polymeric casting compositions UCB, S.A. (BE) 2000-04-18 US disclosed
EP-0810992-A1 SULFUR-CONTAINING COMPOUNDS FOR OPTICAL GRADE POLYMERIC CASTING COMPOSITIONS U C B, S.A. (BE) 1997-12-10 EP disclosed
WO-1996026184-A1 SULFUR-CONTAINING COMPOUNDS FOR OPTICAL GRADE POLYMERIC CASTING COMPOSITIONS UCB, S.A. (BE) 1996-08-29 WO disclosed