SCHEMBL7769823

SCHEMBL7769823

Clc1ccccc1C(c1ccccc1)(c1ccccc1)N1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 3/20 0.48
KCNA3 P22001 2/20 0.48
SLC6A2 P23975 7/20 0.47
SLC6A4 P31645 7/20 0.47
ADRB1 P08588 4/20 0.47
SLC6A3 Q01959 4/20 0.47
CYP1A2 P05177 3/20 0.47
CYP2D6 P10635 3/20 0.47
CYP2C19 P33261 3/20 0.47
CYP2C9 P11712 2/20 0.47
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
CHRM2 P08172 2/20 0.47
CHRM4 P08173 2/20 0.47
CHRM1 P11229 2/20 0.47
CHRM3 P20309 2/20 0.47
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
OPRK1 P41145 2/20 0.47
KCNH2 Q12809 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15587141 0.91 KCNN4 (0.46) KCNN4KCNA3SLC6A2SLC6A4ADRB1
SCHEMBL569963 0.82 SIGMAR1 (0.48) ADRB1CYP1A2CYP2D6CHRM2CHRM4
SCHEMBL8411629 0.81 SIGMAR1 (0.47) ADRB1CYP1A2CYP2D6CHRM2CHRM4
SCHEMBL9090858 0.81 SIGMAR1 (0.47) ADRB1CYP1A2CYP2D6CHRM2CHRM4
SCHEMBL5280949 0.81 KCNN4 (0.48) KCNN4KCNA3SLC6A2SLC6A4ADRB1
SCHEMBL2491431 0.81 ADRB1 (0.49) SLC6A2SLC6A4ADRB1CYP1A2CYP2D6
SCHEMBL2491597 0.81 CHRM2 (0.40) SLC6A2SLC6A4ADRB1SLC6A3CYP2D6
SCHEMBL7336645 0.79 HTR7 (0.49) ADRB1CYP1A2CHRM2CHRM4CHRM1
SCHEMBL7777404 0.78 KCNN4 (0.46) KCNN4KCNA3SLC6A2SLC6A4ADRB1
SCHEMBL2490245 0.77 HTR3A (0.49) SLC6A2SLC6A4ADRB1SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574906-B1 Piperazine and homopiperazine derivatives, pharmaceutical compositions containing them and process for preparing the same NISSHIN FLOUR MILLING CO (JP) 2001-08-22 EP disclosed
US-5380724-A Inhibitors of lipid peroxidation GYOGYSZERKUTATO INTEZET KFT (HU) 1995-01-10 US disclosed
EP-0574906-A2 Piperazine and homopiperazine derivatives, pharmaceutical compositions containing them and process for preparing the same NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-12-22 EP disclosed