SCHEMBL7780419

SCHEMBL7780419

COc1ccc(C(NC(C)c2ccc(F)c(F)c2)c2cccc(N)c2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 1/20 0.43
SOS1 Q07889 1/20 0.43
ACHE P22303 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CASR P41180 2/20 0.38
KDM1A O60341 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
GAA P10253 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785127 0.87 ALDH1A1 (0.41) KRASSOS1ACHECA1CA2
SCHEMBL7780432 0.87 ALDH1A1 (0.41) KRASSOS1ACHECA1CA2
SCHEMBL7780640 0.87 ALDH1A1 (0.41) KRASSOS1ACHECA1CA2
SCHEMBL27553525 0.85 PDPK1 (0.39) KRASSOS1CASRSMN1; SMN2TDP1
SCHEMBL7784936 0.85 PDPK1 (0.39) KRASSOS1CASRSMN1; SMN2TDP1
SCHEMBL7780509 0.84 MAPKAPK2 (0.34) KRASSOS1L3MBTL1ALDH1A1KMT2A
SCHEMBL7785234 0.84 MAPKAPK2 (0.34) KRASSOS1L3MBTL1ALDH1A1KMT2A
SCHEMBL7784937 0.84 KRAS (0.37) KRASSOS1ACHECA1CA2
SCHEMBL7780705 0.83 LMNA (0.34) KRASSOS1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL7785101 0.83 ADRB2 (0.36) KRASSOS1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed