SCHEMBL7780668

SCHEMBL7780668

COc1cc(C(=O)N(C)c2ccccc2OCCCCCC(=O)N2CCN(C)CC2)ccc1NC(=O)c1ccccc1NCCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
POLB P06746 1/20 0.44
AVPR2 P30518 4/20 0.43
AVPR1A P37288 4/20 0.43
AVPR1B P47901 4/20 0.43
KMT2A Q03164 3/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAP3K7 O43318 3/20 0.39
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DRD2 P14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008232 0.93 ALDH1A1 (0.47) ALDH1A1POLBAVPR2AVPR1AAVPR1B
SCHEMBL7339504 0.88 AVPR2 (0.43) ALDH1A1POLBAVPR2AVPR1AAVPR1B
SCHEMBL7374171 0.86 AVPR2 (0.56) AVPR2AVPR1AAVPR1B
SCHEMBL7780700 0.86 AVPR2 (0.48) ALDH1A1POLBAVPR2AVPR1AAVPR1B
SCHEMBL7743965 0.86 AVPR2 (0.52) AVPR2AVPR1AAVPR1B
SCHEMBL8611049 0.85 ALDH1A1 (0.44) ALDH1A1POLBAVPR2AVPR1AAVPR1B
SCHEMBL7344704 0.85 AVPR2 (0.45) AVPR2AVPR1AAVPR1BKMT2AMEN1
SCHEMBL7780670 0.85 KMT2A (0.40) ALDH1A1POLBKMT2AMEN1LMNA
SCHEMBL7778671 0.85 ALDH1A1 (0.44) ALDH1A1POLBAVPR2AVPR1AAVPR1B
SCHEMBL7338041 0.85 AVPR2 (0.42) ALDH1A1POLBAVPR2AVPR1AAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed