SCHEMBL7785401

SCHEMBL7785401

Nc1nc(CO/N=C\C(=O)Oc2cccc3sc(S)nc23)cs1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.34
CYP3A4 P08684 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TP53 P04637 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRB2 P47870 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
NPC1 O15118 3/20 0.31
RAB9A P51151 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3132616 1.00 ALDH1A1 (0.36) ALDH1A1MAPTCYP3A4TDP1TP53
SCHEMBL2789164 0.71 GABRA5 (0.51) ALDH1A1MAPTTP53HTTNPSR1
SCHEMBL3999942 0.71 GABRA5 (0.51) ALDH1A1MAPTTP53HTTNPSR1
SCHEMBL4824847 0.71 GABRA5 (0.47) ALDH1A1MAPTTP53HTTNPSR1
SCHEMBL8940333 0.70 ALDH1A1 (0.39) ALDH1A1MAPTCYP3A4HTTNPSR1
SCHEMBL8896790 0.70 NPC1 (0.47) ALDH1A1MAPTTDP1HTTGABRA5
SCHEMBL8896803 0.70 NPC1 (0.47) ALDH1A1MAPTTDP1HTTGABRA5
Hydrochloric Acid SCHEMBL8913011 0.70 GABRA5 (0.50) ALDH1A1MAPTTP53HTTNPSR1
SCHEMBL4731844 0.69 TDP1 (0.39) ALDH1A1MAPTCYP3A4TDP1NPC1
SCHEMBL1583122 0.69 TDP1 (0.39) ALDH1A1MAPTCYP3A4TDP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640608-B1 Intermediates in the synthesis of cephalosporins BIOCHEMIE GMBH (AT) 2001-11-28 EP disclosed
US-5639877-A AMIDINE SALT OF 7-AMINO-3-HYDROXYMETHYL-3-CEPHEM-4-CARBOXYLIC ACID BIOCHEMIE GESELLSCHAFT M.B.H. (AT) 1997-06-17 US disclosed
EP-0640608-A1 Intermediates in the synthesis of cephalosporins BIOCHEMIE GESELLSCHAFT M.B.H. (AT) 1995-03-01 EP disclosed