SCHEMBL7787012

SCHEMBL7787012

Cc1cc(C(=O)NC(CO)Cc2ccccc2)ccc1-c1ccc2ccccc2c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.47
ROCK1 Q13464 4/20 0.47
MAPK1 P28482 2/20 0.45
RPS6KA5 O75582 1/20 0.45
RPS6KA4 O75676 1/20 0.45
PRKACA P17612 1/20 0.45
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
IRAK1 P51617 1/20 0.45
PRKX P51817 1/20 0.45
PRKG1 Q13976 1/20 0.45
PKN2 Q16513 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
SGK2 Q9HBY8 1/20 0.45
DYRK1A Q13627 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
PIN1 Q13526 5/20 0.45
MME P08473 1/20 0.44
BACE1 P56817 1/20 0.44
DGAT2 Q96PD7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787042 0.87 DYRK1A (0.47) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7787789 0.86 CAPN1 (0.48) PIN1
SCHEMBL7782141 0.85 HPGDS (0.47) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7782210 0.84 DYRK1A (0.47) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7790079 0.83 ROCK2 (0.43) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7786982 0.79 ROCK2 (0.50) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7314496 0.79 PIN1 (0.48) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7322390 0.78 ROCK2 (0.42) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL31611825 0.78 ROCK2 (0.60) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4
SCHEMBL7789971 0.77 DYRK1A (0.44) ROCK2ROCK1MAPK1RPS6KA5RPS6KA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed