SCHEMBL7786982

SCHEMBL7786982

NC(=O)c1c(Cc2ccc(C(=O)NC(CO)Cc3ccccc3)cc2)ccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.50
ROCK1 Q13464 4/20 0.50
PRKACA P17612 2/20 0.50
IRAK1 P51617 2/20 0.50
PRKX P51817 2/20 0.50
PRKG1 Q13976 2/20 0.50
PKN2 Q16513 2/20 0.50
CLK4 Q9HAZ1 2/20 0.50
MAPK1 P28482 2/20 0.50
RPS6KA5 O75582 1/20 0.50
RPS6KA4 O75676 1/20 0.50
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
SGK2 Q9HBY8 1/20 0.50
PIN1 Q13526 5/20 0.44
CTRB1 P17538 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KMT2A Q03164 1/20 0.43
RPS6KB1 P23443 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314900 0.85 PYGL (0.43) NPC1RAB9APLA2G10PLA2G2A
SCHEMBL7313788 0.85 CAPN1 (0.48) CTSL
SCHEMBL7789995 0.85 CAPN1 (0.54) NPC1RAB9ACTSLPLA2G10PLA2G2A
SCHEMBL28227062 0.80 PLA2G10 (0.46) KMT2APLA2G10PLA2G2A
SCHEMBL7787012 0.79 ROCK2 (0.47) ROCK2ROCK1PRKACAIRAK1PRKX
SCHEMBL7322246 0.79 TSHR (0.50) PLA2G10PLA2G2A
SCHEMBL7782141 0.78 HPGDS (0.47) ROCK2ROCK1PRKACAIRAK1PRKX
SCHEMBL7782210 0.78 DYRK1A (0.47) ROCK2ROCK1PRKACAIRAK1PRKX
SCHEMBL7314496 0.78 PIN1 (0.48) ROCK2ROCK1PRKACAIRAK1PRKX
SCHEMBL7787042 0.78 DYRK1A (0.47) ROCK2ROCK1PRKACAIRAK1PRKX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed