SCHEMBL7789971

SCHEMBL7789971

NC(=O)c1c(-c2cc([N+](=O)[O-])ccc2C(=O)NC(CO)Cc2ccccc2)ccc2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
PIN1 Q13526 2/20 0.43
LMNA P02545 3/20 0.41
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TNF P01375 1/20 0.40
MAPT P10636 1/20 0.40
NOD1 Q9Y239 1/20 0.40
CCR3 P51677 5/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
RPS6KA4 O75676 1/20 0.40
PRKACA P17612 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790034 0.87 CAPN1 (0.48) LMNAMEN1POLBKMT2ANPC1
SCHEMBL7782210 0.86 DYRK1A (0.47) DYRK1ADYRK1BPIN1ROCK2RPS6KA5
SCHEMBL7787034 0.80 ALDH1A1 (0.47) LMNAMEN1POLBKMT2ANPC1
SCHEMBL7787042 0.78 DYRK1A (0.47) DYRK1ADYRK1BPIN1MEN1KMT2A
SCHEMBL7790079 0.78 ROCK2 (0.43) DYRK1ADYRK1BPIN1ROCK2RPS6KA5
SCHEMBL7787012 0.77 ROCK2 (0.47) DYRK1ADYRK1BPIN1ROCK2RPS6KA5
SCHEMBL7782141 0.76 HPGDS (0.47) DYRK1ADYRK1BPIN1ROCK2RPS6KA5
SCHEMBL7786987 0.76 CAPN1 (0.45) DYRK1ADYRK1BPIN1ROCK2RPS6KA5
SCHEMBL7782223 0.74 MEN1 (0.47) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL7380790 0.74 LMNA (0.52) PIN1LMNAMEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed