SCHEMBL7787570

SCHEMBL7787570

C=CCNC(=O)c1cc(Br)ccc1Nc1ccc(I)cc1C.C=CCNC(=O)c1cc(F)ccc1Nc1ccc(I)cc1C.C=CCNC(=O)c1cc([N+](=O)[O-])ccc1Nc1ccc(I)cc1C.Cc1cc(I)ccc1Nc1cc(F)ccc1CO.Cc1cc(I)ccc1Nc1ccc(Br)cc1C(=O)NCc1ccc(S(N)(=O)=O)cc1.Cc1cc(I)ccc1Nc1ccc(F)cc1C(=O)NCc1ccc(S(N)(=O)=O)cc1.Cc1cc(I)ccc1Nc1ccc(I)cc1C(=O)NOCc1ccccc1.Cc1cc(I)ccc1Nc1ccc([N+](=O)[O-])cc1C(=O)NC1CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.33
PTGS2 P35354 1/20 0.31
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7932216 0.96 AKR1C3 (0.31) AKR1C3
SCHEMBL7802511 0.95 AKR1C3 (0.30) AKR1C3
SCHEMBL7787200 0.89 PTGS2 (0.31) AKR1C3PTGS2
SCHEMBL7804341 0.87 CA2 (0.37) LMNAHTTSMN1; SMN2
SCHEMBL7794482 0.84 CA2 (0.38) AKR1C3LMNASMN1; SMN2
SCHEMBL7784784 0.83 MT-CO2 (0.39) AKR1C3LMNASMN1; SMN2
SCHEMBL7938680 0.83 MT-CO2 (0.32)
SCHEMBL7784776 0.82 CA2 (0.43) AKR1C3
SCHEMBL7800347 0.80 MAPT (0.40) AKR1C3PTGS2LMNASMN1; SMN2THRB
SCHEMBL7784773 0.79 MAPT (0.36) AKR1C3PTGS2SMN1; SMN2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140067-A1 ANTIVIRAL METHOD USING MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-10-10 EP disclosed
WO-2000037141-A9 COMBINATION CHEMOTHERAPY WARNER LAMBERT CO (US) 2000-12-07 WO disclosed
WO-2000040237-A1 ANTIVIRAL METHOD USING MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2000-07-13 WO disclosed