SCHEMBL7788754

SCHEMBL7788754

N=C(N)Nc1cccc(S(=O)(=O)Nc2cccc(C(CC(=O)O)NC(=O)c3ccc4ccccc4c3)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.51
ITGA2B P08514 3/20 0.51
GPR27 Q9NS67 1/20 0.47
AKR1C3 P42330 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
PLAU P00749 3/20 0.41
ITGAV P06756 1/20 0.41
ITGA2 P17301 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
AR P10275 1/20 0.40
F2 P00734 3/20 0.40
PRSS1 P07477 2/20 0.40
TMPRSS6 Q8IU80 1/20 0.40
MAPT P10636 1/20 0.40
PLG P00747 1/20 0.40
PLAT P00750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7194908 0.91 ITGB3 (0.51) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7781212 0.90 ITGB3 (0.48) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7786217 0.88 KMT2A (0.46) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7789975 0.88 ITGB3 (0.46) ITGB3ITGA2BMEN1KMT2APLAU
SCHEMBL7790184 0.88 MEN1 (0.48) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7785662 0.87 MAPT (0.48) ITGB3ITGA2BMEN1KMT2AITGA2
SCHEMBL7785609 0.87 LMNA (0.45) ITGB3ITGA2BMEN1KMT2AITGA2
SCHEMBL7786246 0.87 ITGB3 (0.46) ITGB3ITGA2BMEN1KMT2AMAPT
SCHEMBL7790080 0.87 MEN1 (0.52) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7781187 0.86 GAA (0.47) ITGB3ITGA2BMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed