SCHEMBL7789975

SCHEMBL7789975

Cc1ccc(C(=O)NC(CC(=O)O)c2cccc(NS(=O)(=O)c3cccc(NC(=N)N)c3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.46
ITGA2B P08514 1/20 0.46
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
KCNA5 P22460 1/20 0.42
ITGAV P06756 1/20 0.42
CASP3 P42574 1/20 0.41
PKM P14618 1/20 0.40
EGFR P00533 1/20 0.40
FGFR1 P11362 1/20 0.40
KDR P35968 1/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
HPN P05981 2/20 0.40
PLAU P00749 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7194908 0.93 ITGB3 (0.51) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7790080 0.92 MEN1 (0.52) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7781212 0.91 ITGB3 (0.48) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7790184 0.91 MEN1 (0.48) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7785662 0.91 MAPT (0.48) ITGB3ITGA2BMEN1KMT2AMAPT
SCHEMBL7781187 0.90 GAA (0.47) ITGB3ITGA2BMEN1KMT2AKCNA5
SCHEMBL7788290 0.89 ITGB3 (0.43) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7786217 0.88 KMT2A (0.46) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7788754 0.88 ITGB3 (0.51) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7785609 0.87 LMNA (0.45) ITGB3ITGA2BMEN1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed