SCHEMBL6945342

SCHEMBL6945342

CCOC(=O)CC(Cc1ccccc1)NC(=O)c1ccc(NC(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 7/20 0.55
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
NR1H4 Q96RI1 1/20 0.51
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
CASP3 P42574 2/20 0.50
SENP7 Q9BQF6 2/20 0.50
SMN1; SMN2 Q16637 3/20 0.48
GAA P10253 1/20 0.48
DEGS1 O15121 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 2/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
DGAT1 O75907 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946318 0.87 PIN1 (0.66) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL7789871 0.83 PIN1 (0.60) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL7789870 0.83 PIN1 (0.60) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL6941033 0.82 CA12 (0.55) PIN1CA12CA1CA2CA9
SCHEMBL11639538 0.81 RAB9A (0.57) PIN1CA2KMT2ANPC1RAB9A
SCHEMBL7789989 0.76 NR1H4 (0.58) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL7789992 0.76 NR1H4 (0.58) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL7781982 0.76 RAB9A (0.72) CA12CA1CA2CA9MEN1
SCHEMBL7782138 0.75 NPC1 (0.59) PIN1MEN1KMT2ANR1H4NPC1
SCHEMBL7322390 0.75 ROCK2 (0.42) PIN1RAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944582-B1 KETOBENZAMIDES AS CALPAIN INHIBITORS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
US-6103720-A ENZYME INHIBITORS; ANTIICHEMIC AND -TUMOR AGENTS; STROKES; ALZEIMER'S DISEASE BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed
EP-0944582-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998025883-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-18 WO disclosed