SCHEMBL7790683

SCHEMBL7790683

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)Oc1ccc(CCC(=O)O)cc1OC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C.CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)Oc1ccc(CCC(=O)OCCl)cc1OC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.46
CA1 P00915 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
CTSL P07711 3/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CTSD P07339 1/20 0.41
FFAR1 O14842 1/20 0.41
CASP3 P42574 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CAPN1 P07384 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3740295 0.97 CASP1 (0.46) CASP1CA1CA2CA5ACTSL
SCHEMBL3734188 0.92 FFAR4 (0.49) CASP1CA1FFAR4CA2CA5A
SCHEMBL3727193 0.86 CTSD (0.49) CASP1CA1CA2CA5ACTSL
SCHEMBL7787410 0.85 CASP1 (0.44) CASP1CA1CA2CA5ACTSL
SCHEMBL3728055 0.84 CTSL (0.53) CASP1FFAR4CTSLCTSBCTSS
SCHEMBL7787424 0.82 CTSD (0.49) CTSLCTSBCTSSCTSKMEN1
SCHEMBL3740038 0.79 CTSL (0.50) CA2CA5ACTSLCTSBCTSS
SCHEMBL7791790 0.79 CTSL (0.48) CASP1CA1CTSLCTSBCTSS
SCHEMBL7791929 0.79 CTSD (0.44) CASP1CTSLCTSSCTSKCTSD
SCHEMBL3725680 0.78 CTSB (0.51) CA2CA5ACTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150956-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MEDIVIR AB (SE) 2001-11-07 EP disclosed
WO-2000047561-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MEDIVIR AB (SE) 2000-08-17 WO disclosed