SCHEMBL7798409

SCHEMBL7798409

COc1ccc(C(C)N)cc1OC.O=C(O)c1ccc(-c2ccccc2)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.44
AKR1C2 P52895 3/20 0.44
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
CASR P41180 2/20 0.42
PDE4A P27815 4/20 0.40
PDE4B Q07343 4/20 0.40
PDE4C Q08493 4/20 0.40
PDE4D Q08499 4/20 0.40
ALDH1A1 P00352 1/20 0.40
ERN1 O75460 1/20 0.40
TRIM24 O15164 1/20 0.40
TRIM33 Q9UPN9 1/20 0.40
LTB4R Q15722 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7792608 0.90 HPGD (0.46) AKR1C3AKR1C2RXRARXRBRXRG
SCHEMBL7798808 0.86 ALDH1A1 (0.45) AKR1C3AKR1C2CASRALDH1A1CA1
SCHEMBL7798405 0.82 SMN1; SMN2 (0.46) RXRARXRBRXRGPDE4APDE4B
SCHEMBL7798400 0.80 HDAC1 (0.43) RXRARXRBRXRGPDE4APDE4B
SCHEMBL8035858 0.74 MAOB (0.46) RXRARXRBRXRGTRIM24TRIM33
SCHEMBL8035116 0.73 PTGES (0.48) RXRARXRBRXRGALDH1A1TRIM24
Phenethylamine SCHEMBL7799179 0.72 RXRA (0.52) RXRARXRBRXRGALDH1A1TRIM24
4-Methylbenzoic Acid SCHEMBL7798453 0.72 KDM4E (0.46) ALDH1A1SMN1; SMN2
SCHEMBL7792606 0.72 KDM4E (0.45) RXRARXRBRXRGALDH1A1CA12
4-Methylbenzoic Acid SCHEMBL7798452 0.70 GAA (0.43) ALDH1A1CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed