SCHEMBL7798400

SCHEMBL7798400

CCNc1ccc(OC)c(OC)c1.O=C(O)c1ccc(-c2ccccc2)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
MCHR1 Q99705 5/20 0.42
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ERN1 O75460 1/20 0.41
LTB4R Q15722 3/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Methylbenzoic Acid SCHEMBL7798452 0.91 GAA (0.43) HDAC1HDAC2NPC1GAAMAPT
SCHEMBL7792603 0.90 MAPT (0.44) HDAC1HDAC2NPC1GAAMAPT
SCHEMBL7798805 0.86 CYP1A2 (0.46) HDAC1HDAC2GAAMAPTSMN1; SMN2
SCHEMBL7798405 0.81 SMN1; SMN2 (0.46) RXRARXRBRXRGMAPTSMN1; SMN2
SCHEMBL7798409 0.80 AKR1C3 (0.44) RXRARXRBRXRGSMN1; SMN2ERN1
SCHEMBL8035858 0.74 MAOB (0.46) RXRARXRBRXRGNPC1RAB9A
SCHEMBL8035116 0.72 PTGES (0.48) HDAC1RXRARXRBRXRGMAPT
Phenethylamine SCHEMBL7799179 0.72 RXRA (0.52) RXRARXRBRXRGNPC1RAB9A
4-Methylbenzoic Acid SCHEMBL7798453 0.72 KDM4E (0.46) NPC1GAAMAPTRAB9ASMN1; SMN2
SCHEMBL7792606 0.71 KDM4E (0.45) RXRARXRBRXRGNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed