SCHEMBL7790490

SCHEMBL7790490

COc1ccc([N][C@H]2CC[C@H](O)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
MMP2 P08253 2/20 0.39
MMP3 P08254 2/20 0.39
MMP13 P45452 2/20 0.39
GRM3 Q14832 1/20 0.38
ALDH1A1 P00352 4/20 0.38
SLC18A3 Q16572 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7794037 0.83 CA12 (0.44) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL7793328 0.79 HTR3E (0.38) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL7784589 0.76 HTR3E (0.38) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL13446559 0.75 RAB9A (0.49) ALDH1A1MAPTTSHRSMN1; SMN2RAB9A
SCHEMBL1966687 0.75 RAB9A (0.49) ALDH1A1MAPTTSHRSMN1; SMN2RAB9A
SCHEMBL1966690 0.75 RAB9A (0.49) ALDH1A1MAPTTSHRSMN1; SMN2RAB9A
SCHEMBL8744137 0.74 NOS3 (0.42) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL1506578 0.72 ESR2 (0.59) CA12CA1CA2CA7CA9
SCHEMBL1506422 0.72 ESR2 (0.59) CA12CA1CA2CA7CA9
SCHEMBL1506423 0.72 ESR2 (0.59) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed