SCHEMBL7794042

SCHEMBL7794042

O[C@H]1CC[C@H]([N]c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.40
ITGAV P06756 1/20 0.40
TSHR P16473 5/20 0.35
HSD17B10 Q99714 2/20 0.35
GAA P10253 2/20 0.35
AGTR1 P30556 1/20 0.35
TP53 P04637 1/20 0.34
MAP3K14 Q99558 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.32
NOTUM Q6P988 1/20 0.32
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32
USP2 O75604 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
CASP1 P29466 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7794564 0.84 TSHR (0.41) ITGB3ITGAVTSHRHSD17B10GAA
SCHEMBL7790502 0.79 HTR3E (0.41) TSHRTP53MEN1KMT2AMAPT
SCHEMBL7784589 0.74 HTR3E (0.38) MAPTLMNARAB9ASMN1; SMN2ALDH1A1
SCHEMBL7794544 0.72 HTR3E (0.44) TSHRMEN1KMT2AMAPTLMNA
SCHEMBL7790531 0.71 HTR3E (0.38) ITGB3ITGAVTSHRMEN1KMT2A
SCHEMBL7790021 0.70 HTR3E (0.43) ITGB3ITGAVHSD17B10KMT2AMAPT
SCHEMBL11369080 0.67 ITGB3 (0.58) ITGB3ITGAVTSHRHSD17B10GAA
SCHEMBL7794045 0.66 RAB9A (0.48) MEN1KMT2AMAPTLMNARAB9A
SCHEMBL22581721 0.64 NOTUM (0.58) MEN1KMT2AMAPTNOTUMLMNA
SCHEMBL30567174 0.64 NOTUM (0.58) MEN1KMT2AMAPTNOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed