SCHEMBL7784589

SCHEMBL7784589

O[C@H]1CC[C@H]([N]c2ccc(Cl)cc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 2/20 0.38
HTR3B O95264 2/20 0.38
HTR3A P46098 2/20 0.38
HTR3D Q70Z44 2/20 0.38
HTR3C Q8WXA8 2/20 0.38
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
SLC22A3 O75751 1/20 0.38
PLAU P00749 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC18A3 Q16572 2/20 0.37
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MAPT P10636 1/20 0.33
CYP1A2 P05177 1/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7793305 0.80 PDE7A (0.41) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7790531 0.80 HTR3E (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7793328 0.80 HTR3E (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7790021 0.79 HTR3E (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794544 0.78 HTR3E (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7790082 0.76 NOS3 (0.42) NPC1RAB9ANOS3NOS1ALDH1A1
SCHEMBL7790490 0.76 NOS3 (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794042 0.74 ITGB3 (0.40) TDP1RAB9AMAPTALDH1A1LMNA
SCHEMBL7784542 0.73 SMN1; SMN2 (0.38) CYP2D6CYP2C19NPC1MAPTLMNA
SCHEMBL7790476 0.73 LMNA (0.46) CYP2C19NPC1RAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed