SCHEMBL7794560

SCHEMBL7794560

COCCC[N]c1ccc(C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ALOX12 P18054 1/20 0.36
KDM4E B2RXH2 1/20 0.36
SCN5A Q14524 2/20 0.35
SCN2A Q99250 2/20 0.35
ACHE P22303 2/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33
SLC22A3 O75751 1/20 0.33
HTR3B O95264 1/20 0.33
PLAU P00749 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7794055 0.77 SCN5A (0.44) SMN1; SMN2NPC1RAB9ASCN5ASCN2A
SCHEMBL11768137 0.74 ACHE (0.39) ALDH1A1SMN1; SMN2NPC1RAB9AACHE
P-Xylene SCHEMBL235090 0.72 ACHE (0.53) ALDH1A1SMN1; SMN2NPC1RAB9AACHE
SCHEMBL8750708 0.72 TDP1 (0.40) ALDH1A1SMN1; SMN2NPC1RAB9ASCN5A
SCHEMBL7789999 0.70 HTR3E (0.43) ALDH1A1SMN1; SMN2NPC1RAB9AACHE
SCHEMBL7793203 0.69 CA1 (0.46) ALDH1A1SMN1; SMN2KDM4EACHEMAPT
SCHEMBL5987245 0.68 DRD2 (0.59) ALDH1A1SMN1; SMN2NPC1KDM4EACHE
SCHEMBL171910 0.68 KCNH2 (0.50) ALDH1A1KDM4ELMNAMAPTCYP2C19
SCHEMBL5985514 0.68 DRD2 (0.59) ALDH1A1SMN1; SMN2NPC1KDM4EACHE
SCHEMBL14232115 0.67 DRD2 (0.57) NPC1KDM4EACHEDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed