SCHEMBL7795285

SCHEMBL7795285

COc1ccc(OC)c(CCc2ccc3ncnc(Cl)c3c2)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 2/20 0.45
ADRA1A P35348 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
P2RX3 P56373 2/20 0.42
ABCB1 P08183 3/20 0.42
AOC3 Q16853 1/20 0.41
DHFR P00374 1/20 0.41
APP P05067 1/20 0.41
EGFR P00533 2/20 0.40
LCK P06239 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803103 0.87 ADRA1A (0.46) ADRA1ATAAR1ALDH1A1LMNAP2RX3
SCHEMBL8439119 0.86 MAP4K4 (0.54) ADRA1ATAAR1P2RX3AOC3DHFR
SCHEMBL4933784 0.85 MTNR1A (0.47) ADRA1ATAAR1P2RX3ABCB1AOC3
SCHEMBL7803101 0.84 CALM1 (0.44) ADRA1ATAAR1ALDH1A1LMNAP2RX3
SCHEMBL7796255 0.82 ADRA1A (0.41) ADRA1ATAAR1P2RX3ABCB1AOC3
SCHEMBL7796168 0.79 MTNR1B (0.43) ALDH1A1P2RX3KMT2A
SCHEMBL29923692 0.79 MAPT (0.56) ENPP1ALDH1A1LMNAEGFRLCK
SCHEMBL591893 0.79 MAPT (0.56) ENPP1ALDH1A1LMNAEGFRLCK
SCHEMBL7796198 0.79 MTNR1A (0.46) ADRA1ATAAR1LMNAP2RX3AOC3
Hydrochloric Acid SCHEMBL28102779 0.77 MAPT (0.55) ENPP1ALDH1A1LMNAEGFRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815087-B1 TRISUBSTITUTED PHENYL DERIVATIVES NOVARTIS AG (CH) 2001-11-14 EP disclosed
US-5990116-A USE IN PREVENTION OR TREATMENT OF INFLAMMATORY AND PROLIFERATIVE SKIN DISEASES AND CANCER; COMPOUNDS SUCH AS 6-(2-(2,5-DIMETHOXYPHENYL)ETHYL)-4-ETHYL-QUINAZOLINE NOVARTIS AG (CH) 1999-11-23 US disclosed
EP-0815087-A1 TRISUBSTITUTED PHENYL DERIVATIVES Novartis AG (CH) 1998-01-07 EP disclosed
WO-1996028430-A1 TRISUBSTITUTED PHENYL DERIVATIVES NOVARTIS AG (CH) 1996-09-19 WO disclosed