SCHEMBL7796022

SCHEMBL7796022

Nc1cccc(Cc2ccc(O)cc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.46
ESR2 Q92731 2/20 0.46
ABAT P80404 1/20 0.43
TAAR1 Q96RJ0 4/20 0.41
SLC6A2 P23975 2/20 0.41
BACE1 P56817 4/20 0.41
KEAP1 Q14145 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
APP P05067 1/20 0.39
BRD4 O60885 1/20 0.38
CD74 P04233 1/20 0.37
MIF P14174 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTR3A P46098 1/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1402167 0.82 BACE1 (0.50) BACE1L3MBTL1APPBRD4ALDH1A1
SCHEMBL29758354 0.82 BACE1 (0.50) BACE1L3MBTL1APPBRD4ALDH1A1
SCHEMBL9395340 0.81 KCNH3 (0.47) TAAR1BACE1L3MBTL1APPNOS3
SCHEMBL28043569 0.81 HSP90AB1 (0.54) SLC6A2BACE1L3MBTL1APPALDH1A1
SCHEMBL28043533 0.79 CYP17A1 (0.47) BACE1L3MBTL1APPNOS3NOS2
SCHEMBL5685326 0.78 ESR1 (0.46) ESR1ESR2ABATTAAR1SLC6A2
SCHEMBL7798261 0.77 ALDH1A1 (0.53) BACE1APPALDH1A1IDO1
SCHEMBL30376292 0.77 TLR8 (0.43) TAAR1BACE1ALDH1A1NOS3NOS2
SCHEMBL28824419 0.74 ADORA2A (0.47) BACE1APPNOS3NOS2
Fumaric Acid SCHEMBL9390245 0.74 LMNA (0.44) BACE1KEAP1BRD4ALDH1A1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010034445-A1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION 2001-10-25 US disclosed
US-6159964-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-12-12 US disclosed
EP-0895475-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2000-08-23 EP disclosed
EP-0906103-A4 1999-04-07 EP disclosed
EP-0906103-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-07 EP disclosed
EP-0895475-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-10 EP disclosed
WO-1997024122-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed
WO-1997024124-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010034445-A1 Vitronectin receptor antagonists ADGRF1, GPR174, CALCRL ESR1 845/4885ESR2 295/4885ABAT 4439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.