SCHEMBL7790129

SCHEMBL7790129

CC(CCC(=O)NCCCC(=O)Cc1cccc(O)c1)CNC(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
SPR P35270 1/20 0.38
CYP3A4 P08684 1/20 0.38
GLS O94925 3/20 0.38
SIRT5 Q9NXA8 1/20 0.37
SIGMAR1 Q99720 2/20 0.36
SYK P43405 1/20 0.36
NQO2 P16083 1/20 0.36
GPR119 Q8TDV5 1/20 0.34
NPFFR1 Q9GZQ6 1/20 0.34
NPFFR2 Q9Y5X5 1/20 0.34
TLR2 O60603 1/20 0.34
TLR1 Q15399 1/20 0.34
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRND Q07001 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796788 0.83 HDAC3 (0.44) SIGMAR1SYK
SCHEMBL7798566 0.73 SYK (0.55) CA1SIRT5SYK
SCHEMBL3715955 0.71 SIGMAR1 (0.56) CA1CA2CYP3A4SIGMAR1SYK
SCHEMBL7799740 0.70 SYK (0.47) SIGMAR1SYK
SCHEMBL7283887 0.70 NQO2 (0.56) CA1CA2SPRCYP3A4SIGMAR1
SCHEMBL7800949 0.70 HDAC3 (0.48) SIGMAR1SYK
SCHEMBL7282857 0.69 NQO2 (0.55) SPRCYP3A4SIGMAR1NQO2
SCHEMBL7799692 0.68 HTT (0.56)
SCHEMBL24815312 0.68 SIGMAR1 (0.58) CA1CA2SIGMAR1NPFFR1NPFFR2
SCHEMBL31505839 0.67 NQO2 (0.62) CA1CA2SPRSIGMAR1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed