SCHEMBL7799437

SCHEMBL7799437

CSc1ccc(C=C(C)C(=O)O)s1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
LIG1 P18858 1/20 0.49
TBXAS1 P24557 2/20 0.44
AKR1C3 P42330 1/20 0.43
APEX1 P27695 8/20 0.41
PLAU P00749 1/20 0.37
PRSS1 P07477 1/20 0.36
TMPRSS15 P98073 1/20 0.36
ERBB2 P04626 1/20 0.35
HTT P42858 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2922217 0.77 MAPT (0.49) PKMTBXAS1AKR1C3APEX1PRSS1
SCHEMBL2922214 0.77 MAPT (0.49) PKMTBXAS1AKR1C3APEX1PRSS1
SCHEMBL9436131 0.71 KMT2A (0.42) PKMLIG1APEX1PLAUERBB2
SCHEMBL7801317 0.71 TBXAS1 (0.43) TBXAS1AKR1C3APEX1PRSS1TMPRSS15
SCHEMBL29088426 0.70 KDM4E (0.47) TBXAS1AKR1C3PRSS1TMPRSS15HTT
SCHEMBL29088392 0.68 PRSS1 (0.41) TBXAS1AKR1C3APEX1PRSS1TMPRSS15
SCHEMBL29088472 0.68 TBXAS1 (0.43) TBXAS1AKR1C3APEX1PRSS1TMPRSS15
SCHEMBL4607795 0.67 DAO (0.41) TBXAS1AKR1C3HTTALDH1A1MAPT
SCHEMBL4607793 0.67 DAO (0.41) TBXAS1AKR1C3HTTALDH1A1MAPT
SCHEMBL9373389 0.66 PKM (0.70) PKMLIG1PLAUALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790245-B1 Substituted Thiophenylalkenylcarbonylguanidide, method for their preparation, their use as medicinal or diagnostic agent as well as medicament containing them HOECHST AG (DE) 2001-06-13 EP claimed