SCHEMBL78001

SCHEMBL78001

CC(C)(C)c1cc(CNCC(F)F)ccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G1B P04054 1/20 0.40
POLB P06746 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
GAA P10253 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
GSR P00390 2/20 0.36
IDO1 P14902 2/20 0.36
DNM1 Q05193 1/20 0.35
KCNH2 Q12809 2/20 0.34
TMEM97 Q5BJF2 2/20 0.34
ANPEP P15144 1/20 0.34
ERAP2 Q6P179 1/20 0.34
P2RX7 Q99572 4/20 0.34
PYCR1 P32322 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MCHR1 Q99705 1/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3085955 0.82 PLA2G1B (0.34) PLA2G1BPOLBATG4BGAACYP1A2
SCHEMBL91286 0.77 POLB (0.40) PLA2G1BPOLBATG4BGAACYP1A2
SCHEMBL3085952 0.72 PLA2G1B (0.33) PLA2G1BPOLBATG4BGAACYP1A2
SCHEMBL19398823 0.71 HSPA5 (0.43) GAACYP1A2CYP2C9CYP2C19IDO1
SCHEMBL3700658 0.71 GAA (0.61) GAACYP2C9CYP2C19DNM1KCNH2
SCHEMBL21674174 0.70 IDO1 (0.53) IDO1P2RX7PYCR1MCHR1HTR1A
SCHEMBL12445277 0.70 IDO1 (0.57) GAACYP1A2CYP2C9CYP2C19IDO1
SCHEMBL26074534 0.70 S1PR1 (0.41) GAACYP1A2CYP2C9CYP2C19GSR
SCHEMBL79109 0.69 P2RX7 (0.50) P2RX7
SCHEMBL2635160 0.69 PRMT5 (0.37) PLA2G1BPOLBATG4BGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed