SCHEMBL7943022

SCHEMBL7943022

NC(=O)N1CCC2(CC1)N=C(N)c1ccccc1N2

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 12/20 0.48
NOS1 P29475 7/20 0.48
NOS3 P29474 2/20 0.48
GAA P10253 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
NEK2 P51955 1/20 0.39
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
KCNH2 Q12809 1/20 0.35
HPGD P15428 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803469 0.88 NOS2 (0.50) NOS2NOS1NOS3GAAALDH1A1
SCHEMBL7804452 0.86 NOS2 (0.57) NOS2NOS1NOS3ALDH1A1NEK2
Hydrochloric Acid SCHEMBL8378262 0.85 NOS2 (0.56) NOS2NOS1NOS3ALDH1A1NEK2
SCHEMBL7803377 0.84 NOS2 (0.55) NOS2NOS1NOS3ALDH1A1NEK2
SCHEMBL7796711 0.84 NOS2 (0.58) NOS2NOS1NOS3NEK2KCNH2
Hydrochloric Acid SCHEMBL8546064 0.84 NOS2 (0.54) NOS2NOS1NOS3ALDH1A1HPGD
SCHEMBL7796668 0.83 NOS2 (0.57) NOS2NOS1NOS3ALDH1A1NEK2
SCHEMBL7931778 0.83 NOS2 (0.57) NOS2NOS1NOS3GAAALDH1A1
SCHEMBL7941207 0.83 NOS2 (0.51) NOS2NOS1NOS3ALDH1A1HPGD
Hydrochloric Acid SCHEMBL8376638 0.83 NOS2 (0.54) NOS2NOS1NOS3ALDH1A1NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed