SCHEMBL7803533

SCHEMBL7803533

COc1nc2ccccc2nc1N(C(=S)Oc1ccccc1)N1CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
HRH4 Q9H3N8 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.33
HTR6 P50406 1/20 0.33
HTR3A P46098 1/20 0.33
HTR2A P28223 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ADRB1 P08588 3/20 0.32
NCF1 P14598 2/20 0.32
ADRB2 P07550 1/20 0.32
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperazine SCHEMBL7803531 0.69 ALDH1A1 (0.35) TP53CYP1A2CYP3A4CYP2D6TSHR
Phenylpiperazine SCHEMBL7795027 0.65 GAA (0.46) TSHRMEN1KMT2AKDM4EHTR3A
SCHEMBL30223071 0.65 HRH4 (0.70) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL24969772 0.65 HRH4 (0.70) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL15195527 0.62 MEN1 (0.47) CYP1A2HRH4MEN1KMT2AKDM4E
SCHEMBL6559651 0.62 L3MBTL1 (0.40) CYP1A2CYP3A4HRH4MEN1KMT2A
SCHEMBL15958678 0.60 EGFR (0.49) MEN1KMT2A
SCHEMBL9216241 0.60 ALDH1A1 (0.62) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL7474377 0.59 NQO2 (0.56) CYP1A2TSHRHRH4MEN1KMT2A
SCHEMBL17295878 0.59 OPRD1 (0.43) CYP2D6TSHRMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075469-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2001-02-14 EP disclosed
WO-2000052001-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-09-08 WO disclosed