SCHEMBL7803748

SCHEMBL7803748

O=CCCc1cc([N+](=O)[O-])ccc1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.54
GPR35 Q9HC97 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CTSB P07858 1/20 0.49
GAA P10253 2/20 0.49
THRB P10828 1/20 0.49
APP P05067 1/20 0.46
NOX4 Q9NPH5 1/20 0.45
CYP1A2 P05177 1/20 0.43
CDC25C P30307 2/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CRHBP P24387 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4006539 0.83 ERN1 (0.57) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL1470136 0.81 TSHR (0.55) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL28013151 0.80 GPR35 (0.53) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL8709893 0.80 THRB (0.56) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL11196837 0.80 CYP1A2 (0.57) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL19742690 0.80 GPR35 (0.53) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL27463698 0.80 SMN1; SMN2 (0.53) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL15283303 0.80 ALDH1A1 (0.56) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL51277 0.79 GPR35 (0.60) ERN1GPR35ALDH1A1TP53HPGD
SCHEMBL11509750 0.78 APP (0.56) ERN1GPR35ALDH1A1TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0956016-A4 PHARMACEUTICAL COMPOUNDS COMPRISING POLYAMINES SUBSTITUTED WITH ELECTRON-AFFINIC GROUPS UNIV FLORIDA STATE (US) 2001-11-14 EP disclosed
US-6255495-B1 KILLING HYPOXIC TUMOR CELLS AND TREATING DERMATOLOGICAL DISEASES IN WARM-BLOODED ANIMALS VIA ADMINISTERING RADIOSENSITIZING AMOUNT OF ELECTRON-AFFINIC-DIAMINE FLORIDA STATE UNIVERSITY 2001-07-03 US disclosed
US-6060604-A FOR RADIOTHERAPY TECHNIQUES, INCREASING TUMOR RADIOSENSITIVITY FLORIDA STATE UNIVERSITY (US) 2000-05-09 US disclosed
US-6057453-A OXIDATION, FORMING RADIOSENSITIZING DIAMINES, REDUCTION FLORIDA STATE UNIVERSITY (US) 2000-05-02 US disclosed
EP-0956016-A1 PHARMACEUTICAL COMPOUNDS COMPRISING POLYAMINES SUBSTITUTED WITH ELECTRON-AFFINIC GROUPS Florida State University (US) 1999-11-17 EP disclosed
CN-1232395-A Pharmaceutical compounds containing polyamines substituted with electron affinity groups UNIV FLORIDA STATE (US) 1999-10-20 CN disclosed
WO-1998014190-A9 PHARMACEUTICAL COMPOUNDS COMPRISING POLYAMINES SUBSTITUTED WITH ELECTRON-AFFINIC GROUPS 1998-07-30 WO disclosed
WO-1998014190-A1 PHARMACEUTICAL COMPOUNDS COMPRISING POLYAMINES SUBSTITUTED WITH ELECTRON-AFFINIC GROUPS FLORIDA STATE UNIVERSITY (US) 1998-04-09 WO disclosed