SCHEMBL7803874

SCHEMBL7803874

Cc1nc(-c2ccccc2)nn1-c1ccccc1OC#CN(C)C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.36
NR1H3 Q13133 4/20 0.35
NR1H2 P55055 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ADORA3 P0DMS8 5/20 0.35
AVPR2 P30518 1/20 0.34
AVPR1A P37288 1/20 0.34
ADORA2A P29274 1/20 0.33
TP53 P04637 1/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561450 0.76 HTR7 (0.50) ADORA1AVPR2AVPR1AMAPTTSHR
SCHEMBL6561418 0.73 BRD4 (0.49) ADORA1NR1H3NPC1RAB9AADORA3
SCHEMBL14118409 0.72 ALDH1A1 (0.50) ADORA1NR1H3NR1H2NPC1RAB9A
SCHEMBL6559724 0.70 GAA (0.47) ADORA1NR1H3NR1H2NPC1RAB9A
SCHEMBL14007393 0.67 NPC1 (0.52) NR1H3NR1H2NPC1RAB9AAVPR1A
SCHEMBL14210107 0.62 NPC1 (0.45) NR1H3NR1H2NPC1RAB9AAVPR1A
SCHEMBL18952840 0.61 NR1H3 (0.48) NR1H3NR1H2NPC1RAB9ATP53
SCHEMBL16202035 0.61 NR1H3 (0.71) NR1H3NR1H2NPC1RAB9AMAPT
SCHEMBL16642051 0.59 TDP2 (0.43) RAB9AHSD17B10MAPTTSHRSMN1; SMN2
SCHEMBL711569 0.59 NPC1 (0.41) NR1H3NR1H2NPC1RAB9AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071670-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-01-31 EP disclosed
WO-1999054314-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed