SCHEMBL7804108

SCHEMBL7804108

COc1cncnc1N1CCN(CCCn2ccc3ccc(Cn4cnnc4)cc32)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.36
TLR7 Q9NYK1 5/20 0.36
TLR9 Q9NR96 3/20 0.36
ACHE P22303 4/20 0.35
BACE1 P56817 4/20 0.35
ABCB1 P08183 1/20 0.35
AURKA O14965 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8033403 0.99 HTR7 (0.36) HTR7TLR7TLR9ACHEBACE1
SCHEMBL7804132 0.86 ACHE (0.35) HTR7TLR7TLR9ACHEBACE1
SCHEMBL7798306 0.86 DRD2 (0.37) HTR7TLR7TLR9ABCB1AURKA
Hydrochloric Acid SCHEMBL8031099 0.86 ACHE (0.35) HTR7TLR7TLR9ACHEBACE1
Hydrochloric Acid SCHEMBL8035086 0.85 DRD2 (0.36) HTR7TLR7TLR9ABCB1AURKA
SCHEMBL7806996 0.84 HTR1A (0.39) HTR7TLR7TLR9ABCB1AURKA
SCHEMBL6999464 0.82 HTR7 (0.41) HTR7MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7803871 0.81 ABCB1 (0.38) TLR7TLR9ABCB1AURKAMEN1
Hydrochloric Acid SCHEMBL6990810 0.81 SLC2A1 (0.41) HTR7MEN1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8035161 0.80 ABCB1 (0.38) HTR7TLR7TLR9ABCB1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed