Scriptaid

Scriptaid

SCHEMBL780490

O=C(CCCCCN1C(=O)c2cccc3cccc(c23)C1=O)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 12/20 1.00
HDAC3 O15379 11/20 1.00
HDAC1 Q13547 11/20 1.00
HDAC11 Q96DB2 11/20 1.00
HDAC6 Q9UBN7 11/20 1.00
HDAC2 Q92769 9/20 1.00
HDAC7 Q8WUI4 8/20 1.00
HDAC10 Q969S8 8/20 1.00
HDAC5 Q9UQL6 8/20 1.00
HDAC4 P56524 7/20 1.00
HDAC9 Q9UKV0 7/20 1.00
NCOR2 Q9Y618 7/20 1.00
ALDH1A1 P00352 6/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
LTA4H P09960 1/20 1.00
KDM4E B2RXH2 5/20 0.73
GAA P10253 1/20 0.73
HTT P42858 1/20 0.73
L3MBTL1 Q9Y468 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Scriptaid SCHEMBL29383029 1.00 HDAC8 (1.00) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL29382031 0.94 ALDH1A1 (0.90) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL411511 0.94 ALDH1A1 (0.90) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL5852563 0.91 HDAC8 (0.83) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL10323380 0.88 ALDH1A1 (0.79) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL14862921 0.87 HDAC8 (1.00) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL30304758 0.87 HDAC8 (1.00) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL19513510 0.87 HDAC1 (0.76) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL20258450 0.85 KDM4E (0.84) HDAC8HDAC3HDAC1HDAC11HDAC6
SCHEMBL18373230 0.85 ALDH1A1 (0.74) HDAC8HDAC3HDAC1HDAC11HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1271 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
WO-2026107052-A1 COMBINATION TREATMENTS USING EPIGENETIC INHIBITION AND SYNGRI-MEDIATED FRATAXIN EXPRESSION ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2026-05-21 WO claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
EP-4720316-A2 NON-VIRAL CELL ENGINEERING Arsenal Biosciences, Inc. (US) 2026-04-08 EP claimed
EP-4673532-A1 THERAPY Plasticell Limited (GB) 2026-01-07 EP claimed
US-12496357-B2 Compositions and methods for treating sickle cell disease YALE UNIVERSITY (US) 2025-12-16 US claimed
US-20250375441-A1 ONCOLYTIC THERAPY WITH A DUAL HDAC3 AND HDAC8 TARGETING AGENT UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2025-12-11 US claimed
EP-3350313-B1 DERIVATION OF LIVER ORGANOIDS FROM HUMAN PLURIPOTENT STEM CELLS AGENCY FOR SCIENCE TECH AND RESEARCH ASTARSTAR (SG) 2025-11-26 EP claimed
US-20250268841-A1 Trans-Epithelial Membrane Drug Delivery System Masiz, John J. (US) 2025-08-28 US claimed
EP-2117536-A2 COSMETIC AND PHARMACEUTICAL APPLICATIONS OF N-ACYLATED AMINO ACIDS AND STRUCTURALLY RELATED COMPOUNDS Beiersdorf AG (DE) 2009-11-18 EP claimed
EP-2114442-A1 HAT ACETYLATION PROMOTERS AND USES OF COMPOSITIONS THEREOF IN PROMOTING IMMUNOGENICITY THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2009-11-11 EP claimed
WO-2008101692-A2 COSMETIC AND PHARMACEUTICAL APPLICATIONS OF N-ACETYLHYDROXYPROLINE BEIERSDORF AG (DE) 2008-08-28 WO claimed
WO-2008101693-A2 COSMETIC AND PHARMACEUTICAL APPLICATIONS OF N-ACYLATED AMINO ACIDS AND STRUCTURALLY RELATED COMPOUNDS BEIERSDORF AG (DE) 2008-08-28 WO claimed
WO-2008090534-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF EXCESSIVE WEIGHT GAIN, REDUCTION OF INAPPROPRIATE EATING BEHAVIOURS AND INHIBITION OF BINGE EATING FOR THE TREATMENT OF OBESITY BERAND LIMITED (IE) 2008-07-31 WO claimed
WO-2008086610-A1 HAT ACETYLATION PROMOTERS AND USES OF COMPOSITIONS THEREOF IN PROMOTING IMMUNOGENICITY THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2008-07-24 WO claimed
WO-2008086612-A1 HAT ACETYLATION PROMOTERS AND USES OF COMPOSITIONS THEREOF IN PROMOTING IMMUNOGENICITY THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2008-07-24 WO claimed
WO-2007049262-A1 Methods and compositions for the promotion of neuronal growth and the treatment of asociality and affective disorders BERAND LIMITED (IE) 2007-05-03 WO claimed
US-20060148684-A1 Use of a histone deacetylase inhibitor for treating muscular dystrophies CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE-CNRS (FR) 2006-07-06 US claimed
US-20010031722-A1 Methods and reagents for facilitating transcription NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-10-18 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12496357-B2 Compositions and methods for treating sickle cell disease HBB, HBG1, HBZ HDAC8 4661/4885HDAC3 4845/4885HDAC1 4862/4885
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES WNT3A, GSK3B, GSK3A HDAC8 19/4885HDAC3 97/4885HDAC1 71/4885
US-12605345-B2 Transdermal drug delivery system FABP2, VEGFA, CUTA HDAC8 555/4885HDAC3 2450/4885HDAC1 2024/4885
US-20250375441-A1 ONCOLYTIC THERAPY WITH A DUAL HDAC3 AND HDAC8 TARGETING AGENT HDAC8, HDAC1, HDAC3 HDAC8 1/4885HDAC3 3/4885HDAC1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.