SCHEMBL7805486

SCHEMBL7805486

COc1ccc(COC(=O)N2C[C@@H](SC(c3ccccc3)(c3ccccc3)c3ccccc3)C[C@H]2CO)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
KIF11 P52732 3/20 0.40
TP53 P04637 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
FABP7 O15540 1/20 0.39
FABP5 Q01469 1/20 0.39
BCL9 O00512 1/20 0.39
CTNNB1 P35222 1/20 0.39
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
HCRTR2 O43614 1/20 0.38
AGTR2 P50052 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7805571 0.91 KIF11 (0.40) P2RX4ALDH1A1NPSR1KIF11TP53
Acetic Acid SCHEMBL7809331 0.90 ALDH1A1 (0.39) P2RX4ALDH1A1NPSR1KIF11TP53
SCHEMBL7809176 0.88 HCRTR2 (0.41) P2RX4ALDH1A1NPSR1KIF11TP53
SCHEMBL7806847 0.87 POLB (0.38) P2RX4ALDH1A1NPSR1TP53MMP9
SCHEMBL7811618 0.86 ALDH1A1 (0.42) P2RX4ALDH1A1NPSR1KIF11TP53
SCHEMBL7805543 0.85 TDP1 (0.43) ALDH1A1
SCHEMBL7805536 0.84 CA1 (0.43) ALDH1A1NPSR1TP53MMP1MMP3
SCHEMBL7800320 0.84 MMP1 (0.38) P2RX4ALDH1A1NPSR1KIF11TP53
SCHEMBL7805587 0.83 CHRM1 (0.38) P2RX4ALDH1A1NPSR1KIF11TP53
SCHEMBL7805589 0.83 CHRM1 (0.38) P2RX4ALDH1A1NPSR1KIF11TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed