SCHEMBL7809863

SCHEMBL7809863

COc1ccc2cc(C(O)c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)ccc2c1.COc1ccc2cc(C(OC(C)C)c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)ccc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.36
AKR1C3 P42330 3/20 0.36
AKR1C2 P52895 3/20 0.36
PTGS1 P23219 2/20 0.36
TSHR P16473 2/20 0.36
CDC42 P60953 1/20 0.36
RAC1 P63000 1/20 0.36
CYP1A2 P05177 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36
ABCB11 O95342 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 2/20 0.34
RECQL P46063 1/20 0.34
SIRT2 Q8IXJ6 2/20 0.33
IDH1 O75874 2/20 0.33
ACSS2 Q9NR19 1/20 0.33
ALOX5 P09917 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748920 0.94 PTGS2 (0.38) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL5682208 0.91 AKR1C3 (0.40) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL5749684 0.85 AKR1C3 (0.37) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL7817690 0.84 AKR1C3 (0.36) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL7817687 0.83 LMNA (0.36) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL5678248 0.81 AKR1C3 (0.44) AKR1C3AKR1C2L3MBTL1LMNASIRT2
SCHEMBL7809865 0.80 ACSS2 (0.33) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL7260656 0.79 CA12 (0.36) SIRT2
SCHEMBL5751662 0.79 ALOX5 (0.44) TSHRLMNASIRT2ACSS2ALOX5
SCHEMBL7169255 0.74 SIRT2 (0.40) AKR1C3AKR1C2PTGS1SIRT2ACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073640-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2001-02-07 EP disclosed
WO-1999054309-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-28 WO disclosed