SCHEMBL7811591

SCHEMBL7811591

C=CCOC(=O)N1C[C@H](OS(C)(=O)=O)C[C@H]1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.45
CYP19A1 P11511 1/20 0.36
ALDH1A1 P00352 3/20 0.34
CASP3 P42574 1/20 0.34
FAAH O00519 3/20 0.33
POLB P06746 1/20 0.33
MGLL Q99685 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
F2 P00734 1/20 0.33
ELANE P08246 1/20 0.33
CTSG P08311 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
MMP2 P08253 1/20 0.32
ANPEP P15144 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CHRM1 P11229 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4303297 0.84 ALDH1A1 (0.38) NPSR1ALDH1A1ADRB2ADRB1ADRB3
SCHEMBL3952747 0.83 BRD4 (0.39)
SCHEMBL7807928 0.83 BRD4 (0.39)
SCHEMBL7805526 0.81 CASP3 (0.41) ALDH1A1CASP3POLBMMP2TDP1
SCHEMBL9031817 0.80 NPSR1 (0.33) NPSR1CYP19A1
SCHEMBL7811563 0.80 NPSR1 (0.46) NPSR1CYP19A1ALDH1A1CASP3FAAH
SCHEMBL7805583 0.79 TDP1 (0.40) ALDH1A1TDP1
SCHEMBL7807951 0.79 CYP19A1 (0.32) CYP19A1SIGMAR1MMP2ANPEP
SCHEMBL8832726 0.78 LMNA (0.36) CYP19A1ALDH1A1FAAHPOLBMGLL
SCHEMBL9210982 0.78 LMNA (0.36) CYP19A1ALDH1A1FAAHPOLBMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed