SCHEMBL7817640

SCHEMBL7817640

O=C(O)C(=O)CC(=O)c1ccc(OCc2ccc(F)c(F)c2)s1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 6/20 0.46
FEN1 P39748 6/20 0.46
MAOB P27338 2/20 0.42
MAOA P21397 1/20 0.42
PTPN1 P18031 3/20 0.40
PPARA Q07869 2/20 0.39
RNASEH1 O60930 1/20 0.39
KDM5A P29375 2/20 0.39
KDM5B Q9UGL1 2/20 0.39
KDM4C Q9H3R0 1/20 0.39
F9 P00740 1/20 0.36
F10 P00742 1/20 0.36
FFAR1 O14842 1/20 0.36
MME P08473 1/20 0.36
ACE P12821 1/20 0.36
CPA1 P15085 1/20 0.36
ACE2 Q9BYF1 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7826615 0.86 ERCC5 (0.48) ERCC5FEN1MAOBPTPN1RNASEH1
SCHEMBL7830115 0.84 NR4A2 (0.47) ERCC5FEN1MAOBMAOAPTPN1
SCHEMBL7828346 0.82 ERCC5 (0.55) ERCC5FEN1PTPN1RNASEH1
SCHEMBL6946999 0.73 PTPN1 (0.73) ERCC5FEN1MAOBMAOAPTPN1
SCHEMBL7828114 0.72 ERCC5 (0.49) ERCC5FEN1PTPN1RNASEH1
SCHEMBL7818349 0.66 ERCC5 (0.51) ERCC5FEN1PTPN1RNASEH1
SCHEMBL7077348 0.66 AGTR1 (0.47) F10
SCHEMBL9508267 0.66 ALDH1A1 (0.50) MAOBMAOA
SCHEMBL7081312 0.65 MAOB (0.54) MAOBMAOAFFAR1
SCHEMBL6947084 0.65 PTPN1 (0.70) ERCC5FEN1PTPN1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP claimed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US claimed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP claimed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP disclosed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US disclosed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP disclosed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed