SCHEMBL7818253

SCHEMBL7818253

CC(=O)c1ccc(N(Cc2ccc(F)cc2)Cc2ccc(F)cc2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
RIPK1 Q13546 2/20 0.39
GSK3B P49841 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TRPA1 O75762 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ACKR3 P25106 1/20 0.37
MCHR1 Q99705 1/20 0.37
MAOB P27338 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
HSD17B1 P14061 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832388 0.84 CRHBP (0.44) GSK3BSMN1; SMN2NPC1RAB9ALMNA
SCHEMBL4677165 0.74 DAO (0.44) MEN1KMT2ANPC1RAB9ATAS2R14
SCHEMBL754372 0.73 ALDH1A1 (0.45) ALDH1A1GSK3BSMN1; SMN2MEN1KMT2A
SCHEMBL7818151 0.72 GSK3B (0.44) ALDH1A1GSK3BSMN1; SMN2NPC1RAB9A
SCHEMBL7818275 0.71 HDAC4 (0.45) ALDH1A1GSK3BMEN1KMT2ANPC1
SCHEMBL7828343 0.70 GSK3B (0.42) ALDH1A1GSK3BSMN1; SMN2NPC1RAB9A
SCHEMBL7081312 0.70 MAOB (0.54) ALDH1A1GSK3BSMN1; SMN2MEN1KMT2A
SCHEMBL13992634 0.68 NPC1 (0.75) ALDH1A1SMN1; SMN2MEN1KMT2ANPC1
SCHEMBL6078000 0.68 LMNA (0.55) ALDH1A1RIPK1SMN1; SMN2MEN1KMT2A
SCHEMBL6353625 0.67 HDAC3 (0.47) ALDH1A1SMN1; SMN2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP disclosed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US disclosed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP disclosed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed