SCHEMBL66292

SCHEMBL66292

CCOC(=O)C1=C(OS(=O)(=O)C(F)(F)F)CCN(C(=O)O)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78185 0.86 PDK1 (0.40) ALDH1A1MAPT
SCHEMBL64034 0.73 CHRM5 (0.38) ALDH1A1MAPT
SCHEMBL18586543 0.73 MEN1 (0.37) ALDH1A1MAPTADORA1
SCHEMBL3992432 0.69 ADORA1 (0.37) ALDH1A1MAPTADORA1
SCHEMBL64675 0.69 PDK1 (0.38) ALDH1A1MAPT
SCHEMBL66293 0.68 PPM1B (0.32)
SCHEMBL27097345 0.67 MEN1 (0.36) ALDH1A1MAPTADORA1
SCHEMBL19078526 0.67 ALDH1A1 (0.32) ALDH1A1MAPT
SCHEMBL1082333 0.66 ESR1 (0.39) ALDH1A1MAPTADORA1
SCHEMBL65230 0.66 MAPT (0.33) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed