SCHEMBL7819587

SCHEMBL7819587

N#Cc1c(-c2c(CCCCN)[nH]c3ccccc23)[nH]c(=O)n1-c1cccc([N+](=O)[O-])c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALOX12 P18054 1/20 0.34
ESR1 P03372 1/20 0.34
POLB P06746 2/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
CTSV O60911 1/20 0.34
CTSL P07711 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7819824 0.87 MAPT (0.39) MAPTMEN1KMT2APDE4APDE4B
SCHEMBL7819968 0.79 KMT2A (0.39) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL7821885 0.79 NTRK1 (0.39) MAPTALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL7821934 0.78 PDE9A (0.33) HTR2AHTR2C
SCHEMBL7822940 0.78 CAMK2D (0.38) MAPTKMT2AKDM4EPOLBHTT
SCHEMBL7812544 0.77 NPEPPS (0.38) MEN1KMT2AALDH1A1KDM4ECTSV
Acetic Acid SCHEMBL7840658 0.76 NPEPPS (0.33) ESR1
SCHEMBL7820462 0.74 CAMK2D (0.34) CDK5CDK5R1
SCHEMBL7826410 0.73 CAMK2D (0.33)
Trifluoroacetic Acid SCHEMBL7838986 0.72 SSTR4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP claimed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO claimed