SCHEMBL7819968

SCHEMBL7819968

COc1ccc(-n2c(C#N)c(-c3c(CCCCN)[nH]c4ccccc34)[nH]c2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.39
MEN1 O00255 2/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 4/20 0.38
HSD17B10 Q99714 2/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
RECQL P46063 1/20 0.36
LMNA P02545 3/20 0.36
PTGS1 P23219 1/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA1 P30542 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7821885 0.91 NTRK1 (0.39) MAPTRECQLALDH1A1SMN1; SMN2TDP1
SCHEMBL7822940 0.83 CAMK2D (0.38) KMT2AMAPTPOLBKDM4EADORA3
SCHEMBL7812544 0.82 NPEPPS (0.38) KMT2AMEN1HSD17B10KDM4ELMNA
SCHEMBL7821934 0.81 PDE9A (0.33)
SCHEMBL7819587 0.79 MAPT (0.37) KMT2AMEN1MAPTPOLBKDM4E
Acetic Acid SCHEMBL7840658 0.78 NPEPPS (0.33)
SCHEMBL7820462 0.77 CAMK2D (0.34) TP53
SCHEMBL7827359 0.76 CAMK2D (0.40) KMT2AMEN1MAPTPOLBKDM4E
SCHEMBL7826410 0.76 CAMK2D (0.33)
Trifluoroacetic Acid SCHEMBL7838986 0.75 SSTR4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP disclosed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO disclosed