SCHEMBL7823271

SCHEMBL7823271

N#Cc1c(-c2c(CCCO)[nH]c3ccccc23)[nH]c(=O)n1-c1c[nH]c2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
HPGD P15428 1/20 0.35
PDE9A O76083 4/20 0.34
KDM4E B2RXH2 2/20 0.33
POLB P06746 1/20 0.33
CAMK2D Q13557 1/20 0.33
CDK4 P11802 1/20 0.33
PRKACA P17612 1/20 0.33
PRKACG P22612 1/20 0.33
PRKACB P22694 1/20 0.33
CCND1 P24385 1/20 0.33
PDE1C Q14123 1/20 0.32
IMPDH2 P12268 1/20 0.32
IMPDH1 P20839 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HAT1 O14929 2/20 0.31
EP300 Q09472 2/20 0.31
CBX7 O95931 1/20 0.31
CDYL2 Q8N8U2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7821934 0.90 PDE9A (0.33) PDE9ACAMK2DCDK4PRKACAPRKACG
SCHEMBL7819614 0.88 MPO (0.36) PDE9AKDM4ECAMK2DCDK4PDE1C
SCHEMBL7826355 0.87 ALDH1A1 (0.32) ALDH1A1PDE9A
SCHEMBL7826816 0.86 ALDH1A1 (0.33) ALDH1A1PDE9APOLBMEN1KMT2A
SCHEMBL7819396 0.86 IDO1 (0.33) PDE9AMEN1KMT2A
Trifluoroacetic Acid SCHEMBL7838986 0.84 SSTR4 (0.33) PDE9A
Trifluoroacetic Acid SCHEMBL7839584 0.82 OXER1 (0.30) ALDH1A1
SCHEMBL7820421 0.81 PDE9A (0.40) ALDH1A1HPGDPDE9AKDM4ECDK4
SCHEMBL7812318 0.79 PRKCB (0.33) PDE9AKDM4ECDK4
Trifluoroacetic Acid SCHEMBL7828206 0.75 TPSAB1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP disclosed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO disclosed