SCHEMBL7828031

SCHEMBL7828031

Cc1ccc(NC(=O)CCc2cccc(N)c2)cc1F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.59
CDK8 P49336 1/20 0.57
BACE1 P56817 1/20 0.56
LMNA P02545 3/20 0.55
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 3/20 0.52
RAB9A P51151 1/20 0.52
MAPT P10636 3/20 0.50
GAA P10253 1/20 0.50
TP53 P04637 2/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7839418 0.85 BACE1 (0.54) KMT2ABACE1LMNARAB9AMAPT
SCHEMBL27557775 0.84 BACE1 (0.53) KMT2ACDK8BACE1LMNAMEN1
SCHEMBL1074012 0.81 MAPT (0.68) BACE1RAB9AMAPTGAAALDH1A1
SCHEMBL13501314 0.79 MAPT (0.71) KMT2ALMNARAB9AMAPTGAA
SCHEMBL7827432 0.79 PLAU (0.59) KMT2ABACE1LMNAKDM4EMEN1
SCHEMBL306804 0.78 RAB9A (0.65) KMT2ALMNARAB9AGAAPOLB
SCHEMBL4628541 0.77 MAPT (0.63) LMNARAB9AMAPTGAAALDH1A1
SCHEMBL7841017 0.75 ALDH1A1 (0.55) KMT2ALMNAMEN1RAB9AMAPT
SCHEMBL307284 0.75 POLB (0.51) KMT2ABACE1LMNAMEN1RAB9A
Hydrochloric Acid SCHEMBL8392031 0.75 MAPT (0.77) LMNARAB9AMAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed