SCHEMBL7841017

SCHEMBL7841017

COc1ccc(NC(=O)CCc2cccc(N)c2)cc1Cl

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
MAPT P10636 5/20 0.55
POLB P06746 2/20 0.55
HPGD P15428 1/20 0.54
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
TSHR P16473 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PKM P14618 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306804 0.90 RAB9A (0.65) POLBRAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL7839418 0.86 BACE1 (0.54) ALDH1A1MAPTHPGDRAB9ANPC1
SCHEMBL4666943 0.78 LMNA (0.73) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL14886137 0.78 MAPT (0.67) ALDH1A1MAPTPOLBHPGDMEN1
SCHEMBL306284 0.77 SMN1; SMN2 (0.66) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL2008813 0.77 ALDH1A1 (0.70) ALDH1A1MAPTPOLBHPGDRAB9A
SCHEMBL13501314 0.76 MAPT (0.71) ALDH1A1MAPTHPGDRAB9AKMT2A
SCHEMBL7827432 0.76 PLAU (0.59) ALDH1A1MAPTPOLBHPGDRAB9A
SCHEMBL1074012 0.75 MAPT (0.68) ALDH1A1MAPTPOLBHPGDRAB9A
SCHEMBL7828031 0.75 KMT2A (0.59) ALDH1A1MAPTPOLBRAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed