SCHEMBL7827432

SCHEMBL7827432

Nc1cccc(CCC(=O)Nc2ccc3ccccc3c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.59
CYP1A2 P05177 2/20 0.58
MAPT P10636 4/20 0.57
GAA P10253 2/20 0.57
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
POLB P06746 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
RAB9A P51151 3/20 0.54
LMNA P02545 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NPC1 O15118 1/20 0.54
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP2C19 P33261 1/20 0.52
HIF1A Q16665 1/20 0.52
HDAC1 Q13547 2/20 0.52
HDAC2 Q92769 2/20 0.52
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11628339 0.86 NLRP3 (0.61) CYP1A2MAPTGAAMEN1KMT2A
SCHEMBL28549583 0.86 CYP1A2 (0.72) PLAUCYP1A2MAPTGAAMEN1
SCHEMBL13501314 0.85 MAPT (0.71) MAPTGAAKMT2AL3MBTL1RAB9A
SCHEMBL4628541 0.83 MAPT (0.63) PLAUMAPTGAARAB9ALMNA
SCHEMBL1074012 0.81 MAPT (0.68) PLAUMAPTGAAPOLBRAB9A
SCHEMBL7839198 0.81 RAB9A (0.64) MAPTGAAPOLBRAB9ALMNA
Hydrochloric Acid SCHEMBL8392031 0.81 MAPT (0.77) PLAUMAPTGAAPOLBRAB9A
SCHEMBL7837786 0.79 SENP1 (0.62) MAPTGAARAB9AALDH1A1HDAC1
SCHEMBL7828031 0.79 KMT2A (0.59) MAPTGAAMEN1KMT2APOLB
SCHEMBL306804 0.79 RAB9A (0.65) CYP1A2GAAKMT2APOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed