SCHEMBL7829392

SCHEMBL7829392

N#CC(C#N)c1ncccn1

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.31
MAPT P10636 1/20 0.31
HDAC8 Q9BY41 1/20 0.30
HSP90AA1 P07900 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11877693 0.69 KCNMA1 (0.35)
SCHEMBL11631498 0.67 ALDH1A1 (0.45) ALDH1A1MAPTGAASMN1; SMN2
SCHEMBL27656044 0.66 ALDH1A1 (0.32) ALDH1A1MEN1GAAKMT2ASMN1; SMN2
SCHEMBL86412 0.66 MEN1 (0.44) ALDH1A1MEN1GAAKMT2ASMN1; SMN2
SCHEMBL2541201 0.61
SCHEMBL241029 0.61
SCHEMBL3293919 0.61
SCHEMBL4099364 0.61
SCHEMBL16671626 0.61
SCHEMBL3220940 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274734-B1 Process for making pyrimidine derivatives HOFFMAN-LA ROCHE INC. 2001-08-14 US disclosed
EP-0841326-B1 Process for the preparation of pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2001-05-16 EP disclosed
US-6121447-A STARTING WITH 2-CYANOPYRIMIDINE, WHICH IS PREPARED BY REACTING 2-CHLOROPYRIMIDINE WITH AN ALKALI CYANIDE IN THE PRESENCE OF 1-AZABICYCLO(2,2,2)OCTANE OR 1,4-DIAZABICYCLO(2,2,2)OCTANE HOFFMANN-LA ROCHE INC. (US) 2000-09-19 US disclosed
US-5883254-A CYANATION OF PYRIMIDINES BY REACTING WITH AN ALKALI CYANIDE IN THE PRESENCE OF 1-AZABICYCLO(2,2,2)OCTANE OR 1,4-DIAZABICYCLO(2,2,2)OCTANE HOFFMANN-LA ROCHE INC. (US) 1999-03-16 US disclosed
EP-0841326-A1 Process for the preparation of pyrimidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-05-13 EP disclosed