SCHEMBL7833443

SCHEMBL7833443

Cc1cc2c(CN(C)C)c(O)ccc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.54
KDM4E B2RXH2 8/20 0.49
MAPT P10636 6/20 0.49
TDP1 Q9NUW8 3/20 0.49
ALDH1A1 P00352 9/20 0.47
PKM P14618 1/20 0.47
CYP3A4 P08684 2/20 0.46
GRIN2B Q13224 1/20 0.45
HTR7 P34969 3/20 0.42
HTR6 P50406 3/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
HTR2B P41595 1/20 0.42
HSD17B10 Q99714 4/20 0.41
MAPK1 P28482 3/20 0.41
HTR1D P28221 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623327 0.73 ALDH1A1 (0.53) ADRB2KDM4EMAPTTDP1ALDH1A1
SCHEMBL15373471 0.73 NR1I2 (0.51) KDM4EMAPTALDH1A1HSD17B10MAPK1
SCHEMBL296024 0.70 KEAP1 (0.47) KDM4EMAPTALDH1A1HSD17B10MAPK1
SCHEMBL15704609 0.70 HPGD (0.47) KDM4EMAPTALDH1A1HSD17B10MAPK1
SCHEMBL14319825 0.70 CYP3A4 (0.49) KDM4EMAPTALDH1A1CYP3A4HTR6
SCHEMBL2233005 0.70 ADRB2 (1.00) ADRB2KDM4EMAPTTDP1ALDH1A1
SCHEMBL4424885 0.70 NQO2 (0.57) KDM4EMAPTALDH1A1HSD17B10MAPK1
SCHEMBL17829970 0.69 HTR6 (0.75) KDM4EMAPTALDH1A1CYP3A4HTR7
Hydrochloric Acid SCHEMBL2535761 0.69 ADRB2 (0.97) ADRB2KDM4EMAPTTDP1ALDH1A1
Bromide SCHEMBL8994861 0.69 ADRB2 (0.97) ADRB2KDM4EMAPTTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1344270-A Functionalized heterocycles as chemokine receptor modulators THOUSAND YEARS MEDICAMENTS INC (US) 2002-04-10 CN disclosed
EP-1144415-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2001-10-17 EP disclosed
WO-2000042045-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2000-07-20 WO disclosed