SCHEMBL4623327

SCHEMBL4623327

CN(C)Cc1c(O)ccc2[nH]ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
PKM P14618 1/20 0.53
KDM4E B2RXH2 6/20 0.51
MAPT P10636 3/20 0.51
TDP1 Q9NUW8 2/20 0.51
ADRB2 P07550 1/20 0.49
GRIN2B Q13224 1/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
HSD17B10 Q99714 3/20 0.41
CYP3A4 P08684 2/20 0.41
TSHR P16473 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 1/20 0.40
NPY1R P25929 1/20 0.40
MAPK1 P28482 1/20 0.40
AKT1 P31749 1/20 0.40
HTT P42858 1/20 0.40
GAA P10253 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1993443 0.83 BCHE (0.40) ALDH1A1PKMKDM4EMAPTTDP1
SCHEMBL31543744 0.80 P2RX7 (0.41) ALDH1A1PKMKDM4EHSD17B10GAA
SCHEMBL28017334 0.80 P2RX7 (0.41) ALDH1A1PKMKDM4EHSD17B10GAA
SCHEMBL1400453 0.77 MTNR1A (0.40) ALDH1A1PKMKDM4EKMT2AMEN1
SCHEMBL3617254 0.77 MTNR1A (0.53) ALDH1A1KDM4EMAPTKMT2AMEN1
SCHEMBL8915154 0.76 ALDH1A1 (0.45) ALDH1A1PKMKDM4EMAPTTDP1
SCHEMBL3621271 0.74 ALDH1A1 (0.42) ALDH1A1PKMKDM4EMAPTKMT2A
SCHEMBL7833443 0.73 ADRB2 (0.54) ALDH1A1PKMKDM4EMAPTTDP1
SCHEMBL6804682 0.73 HTR1D (0.36) ALDH1A1PKMKDM4EADRB2HSD17B10
SCHEMBL4624598 0.72 KDM4E (0.51) ALDH1A1PKMKDM4EMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446131-B1 Keratinous fibres dyeing process with substituted monohydroxy indols and compositions OREAL (FR) 1994-05-04 EP claimed
EP-0446131-A1 Keratinous fibres dyeing process with substituted monohydroxy indols and compositions L'OREAL (FR) 1991-09-11 EP claimed
EP-1067950-B1 NEO-TRYPTOPHAN MAYO FOUNDATION (US) 2008-05-14 EP disclosed
CN-1344270-A Functionalized heterocycles as chemokine receptor modulators THOUSAND YEARS MEDICAMENTS INC (US) 2002-04-10 CN disclosed
EP-1144415-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2001-10-17 EP disclosed
WO-2000042045-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2000-07-20 WO disclosed
EP-0446131-B1 Keratinous fibres dyeing process with substituted monohydroxy indols and compositions OREAL (FR) 1994-05-04 EP disclosed
EP-0446131-A1 Keratinous fibres dyeing process with substituted monohydroxy indols and compositions L'OREAL (FR) 1991-09-11 EP disclosed